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O95259 | KCNH1_HUMAN | Potassium voltage-gated channel subfamily H member 1 (KCNH1)

3D structures mapped by conservation among orthologs

[ Domain: "sensor domains" // PAS ]

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[ Alpha Fold Model ] (go)


Known binders annotated in ChEMBL

IC50 table

molecule_chembl_id structure assay_type relation values units mol_wt smiles organism assay_chembl_id bao_label
CHEMBL3261075 OBDepict N N N H O F CH 3 N N H 2 N IC50 = 490.0 nM 388.41 C[C@@]1(c2cc(NC(=O)c3ccc(C#N)cn3)ccc2F)Cn2cccc2C(N)=N1 Homo sapiens CHEMBL4307470 single protein format