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O95398 | RPGF3_HUMAN | Rap guanine nucleotide exchange factor 3 (RAPGEF3)

3D structures mapped by conservation among orthologs



[ Alpha Fold Model ] (go)


Known binders annotated in ChEMBL

IC50 table

molecule_chembl_id structure assay_type relation values units mol_wt smiles organism assay_chembl_id bao_label
CHEMBL4517829 OBDepict CH 3 O S H 2 N HN O O O O O CH 3 IC50 = 900.0 nM 416.46 COc1ccc2ccc(OCC(=O)NS(=O)(=O)c3ccc(N)cc3OC)cc2c1 Homo sapiens CHEMBL4346467 assay format