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P00736 | C1R_HUMAN | Complement C1r subcomponent (C1R)

3D structures mapped by conservation among orthologs

[ Domain: "Spermadhesin, CUB domain" // CUB ]

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[ Domain: "FMN-binding split barrel 2" // Trypsin ]

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[ Domain: "EGF/Laminin" // EGF_CA ]

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[ Domain: "Complement control module/SCR domain" // Sushi ]

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[ Domain: "Complement control module/SCR domain" // Sushi_3 ]

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[ Domain: pdbs with more than 2 multi-domains ]

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[ Alpha Fold Model ] (go)


Known binders annotated in ChEMBL

IC50 table

molecule_chembl_id structure assay_type relation values units mol_wt smiles organism assay_chembl_id bao_label
CHEMBL10770 OBDepict I N H O N O IC50 = 200.0 nM 414.2 O=c1oc(Nc2ccccc2I)nc2cc3ccccc3cc12 Homo sapiens CHEMBL655961 single protein format
CHEMBL10312 OBDepict I N H N O O F F F IC50 = 400.0 nM 432.14 O=c1oc(Nc2ccccc2I)nc2cc(C(F)(F)F)ccc12 Homo sapiens CHEMBL655961 single protein format
CHEMBL10610 OBDepict Cl N O O N H Cl Cl IC50 = 400.0 nM 341.58 O=c1oc(Nc2c(Cl)cccc2Cl)nc2cc(Cl)ccc12 Homo sapiens CHEMBL655961 single protein format
CHEMBL10569 OBDepict I N H N O O Cl Cl IC50 = 500.0 nM 433.03 O=c1oc(Nc2ccccc2I)nc2cc(Cl)c(Cl)cc12 Homo sapiens CHEMBL655961 single protein format
CHEMBL4247936 OBDepict O N H H N O H 3 C CH 3 Cl Cl N H O S HN NH 2 IC50 = 600.0 nM 536.49 CC(C)[C@@H](NC(=O)Cc1c(Cl)cccc1Cl)C(=O)N1CC=CC1C(=O)NCc1ccc(C(=N)N)s1 Homo sapiens CHEMBL4229689 single protein format
CHEMBL10432 OBDepict Cl N O O N H I IC50 = 700.0 nM 398.59 O=c1oc(Nc2ccccc2I)nc2cc(Cl)ccc12 Homo sapiens CHEMBL655961 single protein format
CHEMBL158926 OBDepict I O N O IC50 = 700.0 nM 399.19 O=c1oc(-c2ccccc2I)nc2cc3ccccc3cc12 Homo sapiens CHEMBL655965 single protein format
CHEMBL166801 OBDepict CH 3 O S N O O CH 3 N O O IC50 = 700.0 nM 346.36 COc1ccc(S(=O)(=O)N(C)c2nc3ccccc3c(=O)o2)cc1 Homo sapiens CHEMBL661597 single protein format
CHEMBL10248 OBDepict CH 3 N O O N H I IC50 = 800.0 nM 378.17 Cc1ccc2c(=O)oc(Nc3ccccc3I)nc2c1 Homo sapiens CHEMBL655961 single protein format
CHEMBL10065 OBDepict I N H N O O + N O _ O IC50 = 800.0 nM 409.14 O=c1oc(Nc2ccccc2I)nc2cc([N+](=O)[O-])ccc12 Homo sapiens CHEMBL655961 single protein format
CHEMBL274319 OBDepict Cl N O O N H Cl IC50 = 800.0 nM 307.14 O=c1oc(Nc2ccccc2Cl)nc2cc(Cl)ccc12 Homo sapiens CHEMBL655961 single protein format
CHEMBL10132 OBDepict CH 3 N O O N H Cl IC50 = 900.0 nM 286.72 Cc1ccc2c(=O)oc(Nc3ccccc3Cl)nc2c1 Homo sapiens CHEMBL655960 single protein format
CHEMBL10252 OBDepict Cl N H Cl N O O IC50 = 900.0 nM 307.14 O=c1oc(Nc2c(Cl)cccc2Cl)nc2ccccc12 Homo sapiens CHEMBL655961 single protein format
CHEMBL273264 OBDepict NH 2 HN NH O O NH H 2 N IC50 = 1000.0 nM 347.38 N=C(N)Nc1ccc(C(=O)Oc2ccc3cc(C(=N)N)ccc3c2)cc1 Homo sapiens CHEMBL655965 single protein format