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P01031 | CO5_HUMAN | Complement C5 (C5)

3D structures mapped by conservation among orthologs

[ Domain: "Immunoglobulin/Fibronectin type III/E set domains/PapD-like" // A2M_N_1 ]

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[ Domain: "Common fold of diphtheria toxin/transcription factors/cytochrome f" // A2M_recep ]

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[ Domain: "TIMP-like" // NTR ]

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[ Domain: "Anaphylotoxins (complement system)" // ANATO ]

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[ Domain: "Spermadhesin, CUB domain" // EUF07662 "Immunoglobulin/Fibronectin type III/E set domains/PapD-like" // A2M_N_1 "Common fold of diphtheria toxin/transcription factors/cytochrome f" // A2M_recep "TIMP-like" // NTR "Anaphylotoxins (complement system)" // ANATO ]

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[ Domain: "alpha/alpha toroid" // A2M_comp ]

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[ Domain: "Immunoglobulin/Fibronectin type III/E set domains/PapD-like" // KOG1366_2nd_1 ]

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[ Domain: "Immunoglobulin/Fibronectin type III/E set domains/PapD-like" // ANATO,A2M_N_2 ]

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[ Domain: "Immunoglobulin/Fibronectin type III/E set domains/PapD-like" // MG4 ]

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[ Domain: "Immunoglobulin/Fibronectin type III/E set domains/PapD-like" // KOG1366_1st ]

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[ Domain: "Immunoglobulin/Fibronectin type III/E set domains/PapD-like" // A2M_C ]

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[ Domain: "Immunoglobulin/Fibronectin type III/E set domains/PapD-like" // A2M_N ]

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[ Domain: "Immunoglobulin/Fibronectin type III/E set domains/PapD-like" // A2M_N_2 ]

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[ Domain: pdbs with more than 2 multi-domains ]

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[ Alpha Fold Model ] (go)


Known binders annotated in ChEMBL

IC50 table

molecule_chembl_id structure assay_type relation values units mol_wt smiles organism assay_chembl_id bao_label
CHEMBL4757748 OBDepict CH 3 O O N H N H O CH 3 H 3 C CH 3 H O CH 3 IC50 <= 5.0 nM 400.52 COc1ccc(NC(=O)N[C@@H](C)c2ccccc2OC)cc1OCCCC(C)C Homo sapiens CHEMBL4668571 cell-free format
CHEMBL2203296 OBDepict CH 3 O O NH H 3 C N H O CH 3 H IC50 = 210.0 nM 370.49 CCCCCCOc1cc(NC(=O)N[C@@H](C)c2ccccc2)ccc1OC Homo sapiens CHEMBL4668571 cell-free format
CHEMBL2204196 OBDepict CH 3 O O N H N H O CH 3 H 3 C CH 3 H IC50 = 440.0 nM 370.49 COc1ccc(NC(=O)N[C@@H](C)c2ccccc2)cc1OCCCC(C)C Homo sapiens CHEMBL4668571 cell-free format
CHEMBL4756677 OBDepict CH 3 O O O OH N H N H O H 3 C CH 3 CH 3 H IC50 = 620.0 nM 414.5 COc1cc(C(=O)O)c(NC(=O)N[C@@H](C)c2ccccc2)cc1OCCCC(C)C Homo sapiens CHEMBL4668571 cell-free format