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P11274 | BCR_HUMAN | Breakpoint cluster region protein (BCR)

3D structures mapped by conservation among orthologs

[ Domain: "DBL homology domain (DH-domain)" // RhoGEF ]

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[ Domain: "PH domain-like" // PH_10 ]

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[ Domain: "Bcr-Abl oncoprotein oligomerization domain" // Bcr-Abl_Oligo ]

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[ Domain: pdbs with more than 2 multi-domains ]

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[ Alpha Fold Model ] (go)


Known binders annotated in ChEMBL

IC50 table

molecule_chembl_id structure assay_type relation values units mol_wt smiles organism assay_chembl_id bao_label
CHEMBL434335 OBDepict O NH N H N N H CH 3 CH 3 H 3 C N N N IC50 = 573.0 nM 439.52 Cc1ccc(NC(=O)Nc2cccc(N(C)C)c2)cc1Nc1nccc(-c2cccnc2)n1 Homo sapiens CHEMBL832728 single protein format
CHEMBL184742 OBDepict O NH HN N N H CH 3 N N N IC50 = 720.0 nM 465.56 Cc1ccc(NC(=O)Nc2cccc(N3CCCC3)c2)cc1Nc1nccc(-c2cccnc2)n1 Homo sapiens CHEMBL832728 single protein format