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P14778 | IL1R1_HUMAN | Interleukin-1 receptor type 1 (IL1R1)

3D structures mapped by conservation among orthologs

[ Domain: "Immunoglobulin/Fibronectin type III/E set domains/PapD-like" // I-set_4 ]

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[ Domain: "Immunoglobulin/Fibronectin type III/E set domains/PapD-like" // I-set ]

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[ Domain: "Immunoglobulin/Fibronectin type III/E set domains/PapD-like" // I-set_8 ]

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[ Domain: "Immunoglobulin/Fibronectin type III/E set domains/PapD-like" // I-set_5 ]

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[ Domain: pdbs with more than 2 multi-domains ]

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[ Alpha Fold Model ] (go)


Known binders annotated in ChEMBL

IC50 table

molecule_chembl_id structure assay_type relation values units mol_wt smiles organism assay_chembl_id bao_label
CHEMBL4213787 OBDepict Cl Cl S N N H O N H O N IC50 = 720.0 nM 393.25 O=C(NNC(=O)c1csc(-c2ccc(Cl)cc2Cl)n1)c1ccccn1 Homo sapiens CHEMBL4195489 cell-based format