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P28347 | TEAD1_HUMAN | Transcriptional enhancer factor TEF-1 (TEAD1)

3D structures mapped by conservation among orthologs

[ Domain: "tri-helical" // TEA ]

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[ Domain: "Immunoglobulin/Fibronectin type III/E set domains/PapD-like" // KOG3841 ]

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[ Alpha Fold Model ] (go)


Known binders annotated in ChEMBL

IC50 table

molecule_chembl_id structure assay_type relation values units mol_wt smiles organism assay_chembl_id bao_label
CHEMBL4129172 OBDepict O NH S N N N H IC50 = 83.0 nM 368.51 O=C(CSc1nnc[nH]1)Nc1ccc(C2C3CC4CC(C3)CC2C4)cc1 Homo sapiens CHEMBL4120897 cell-based format