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P40818 | UBP8_HUMAN | Ubiquitin carboxyl-terminal hydrolase 8 (USP8)

3D structures mapped by conservation among orthologs

[ Domain: "Rhodanese/Cell cycle control phosphatase" // UNK_F_TYPE ]

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[ Domain: "Cysteine proteinases" // UCH ]

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[ Domain: "USP8 N-terminal domain-like" // USP8_dimer ]

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[ Alpha Fold Model ] (go)


Known binders annotated in ChEMBL

IC50 table

molecule_chembl_id structure assay_type relation values units mol_wt smiles organism assay_chembl_id bao_label
CHEMBL2398212 OBDepict N N N N O Cl IC50 = 96.0 nM 266.65 N#Cc1nc2c(nc1C#N)-c1ccc(Cl)cc1C2=O Homo sapiens CHEMBL4119760 assay format