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P42568 | AF9_HUMAN | Protein AF-9 (MLLT3)

3D structures mapped by conservation among orthologs

[ Domain: "C2 domain" // YEATS ]

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[ Domain: "Bromodomain-containing protein 4 ET domain" // BET_1 ]

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[ Domain: pdbs with more than 2 multi-domains ]

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[ Alpha Fold Model ] (go)


Known binders annotated in ChEMBL

IC50 table Ki table

molecule_chembl_id structure assay_type relation values units mol_wt smiles organism assay_chembl_id bao_label
CHEMBL4865432 OBDepict F N N NH NH O N N N IC50 = 729.0 nM 377.38 O=C(NCc1ccc(CNc2ncc(F)cn2)cc1)c1ccc2nncn2c1 Homo sapiens CHEMBL4810341 single protein format
CHEMBL4863719 OBDepict O N H N N N N IC50 = 984.0 nM 321.38 O=C(NCc1ccc(CN2CCC2)cc1)c1ccc2nncn2c1 Homo sapiens CHEMBL4810341 single protein format