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Q00532 | CDKL1_HUMAN | Cyclin-dependent kinase-like 1 (CDKL1)

3D structures mapped by conservation among orthologs

[ Domain: "Protein kinase" // Pkinase_Tyr ]

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[ Alpha Fold Model ] (go)


Known binders annotated in ChEMBL

IC50 table

molecule_chembl_id structure assay_type relation values units mol_wt smiles organism assay_chembl_id bao_label
CHEMBL455428 OBDepict CH 3 N H O F NH N N N N CH 3 H 3 C H 3 C IC50 = 60.0 nM 368.42 CNC(=O)c1ccc(Nc2nccc(-c3cnc(C)n3C(C)C)n2)cc1F Homo sapiens CHEMBL1022595 single protein format