Q03164 | KMT2A_HUMAN | Histone-lysine N-methyltransferase 2A (KMT2A)
3D structures mapped by conservation among orthologs
[ Domain: "CXXC domain" // zf-CXXC ]
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[ Domain: "FYVE/PHD zinc finger" // PHD ]
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[ Domain: "Bromodomain" // Bromodomain ]
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[ Domain: "SET domain-like" // SET ]
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[ Alpha Fold Model ] (go)
Known binders annotated in ChEMBL
IC50 table
Ki table
| molecule_chembl_id | structure | assay_type | relation | values | units | mol_wt | smiles | organism | assay_chembl_id | bao_label |
|---|---|---|---|---|---|---|---|---|---|---|
| CHEMBL3798088 | IC50 | = | 320.0 | nM | 586.74 | CC[C@@H]1NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@](C)(NC(=O)C(C)C)CCCCNC(=O)[C@@H](c2ccccc2)NC1=O | Homo sapiens | CHEMBL3801644 | cell-based format |