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Q08188 | TGM3_HUMAN | Protein-glutamine gamma-glutamyltransferase E (TGM3)

3D structures mapped by conservation among orthologs

[ Domain: "Immunoglobulin/Fibronectin type III/E set domains/PapD-like" // Transglut_N ]

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[ Domain: "Immunoglobulin/Fibronectin type III/E set domains/PapD-like" // Transglut_C_1 ]

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[ Domain: "Immunoglobulin/Fibronectin type III/E set domains/PapD-like" // Transglut_C ]

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[ Domain: "Cysteine proteinases" // Transglut_core ]

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[ Domain: pdbs with more than 2 multi-domains ]

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[ Alpha Fold Model ] (go)


Known binders annotated in ChEMBL

IC50 table

molecule_chembl_id structure assay_type relation values units mol_wt smiles organism assay_chembl_id bao_label
CHEMBL2086889 OBDepict CH 3 O N N N H 3 C N O N H 3 C O IC50 = 11.0 nM 313.32 CCn1nc(-c2ccc(OC)cc2)nc2c(=O)n(C)c(=O)nc1-2 Homo sapiens CHEMBL2091159 single protein format