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Q13324 | CRFR2_HUMAN | Corticotropin-releasing factor receptor 2 (CRHR2)

3D structures mapped by conservation among orthologs



[ Alpha Fold Model ] (go)


Known binders annotated in ChEMBL

IC50 table Ki table

molecule_chembl_id structure assay_type relation values units mol_wt smiles organism assay_chembl_id bao_label
CHEMBL3681374 OBDepict H 3 C O Cl N H N H 3 C N H H H N H O Cl F F F IC50 = 727.0 nM 555.43 COc1ccc(-c2c(NC[C@H]3CC[C@H](NC(=O)c4cc(C(F)(F)F)ccc4Cl)CC3)n[nH]c2C)c(Cl)c1 Homo sapiens CHEMBL3707792 cell-based format