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Q13951 | PEBB_HUMAN | Core-binding factor subunit beta (CBFB)

3D structures mapped by conservation among orthologs

[ Domain: "Core binding factor beta, CBF" // CBF_beta ]

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[ Domain: pdbs with more than 2 multi-domains ]

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[ Alpha Fold Model ] (go)


Known binders annotated in ChEMBL

IC50 table

molecule_chembl_id structure assay_type relation values units mol_wt smiles organism assay_chembl_id bao_label
CHEMBL3675784 OBDepict Cl Cl N N H N IC50 = 700.0 nM 264.12 Clc1cc(Cl)c2[nH]c(-c3ccccn3)nc2c1 Homo sapiens CHEMBL3705193 single protein format
CHEMBL3675786 OBDepict Cl N N H F F F N IC50 = 760.0 nM 297.67 FC(F)(F)c1cc(Cl)c2[nH]c(-c3ccccn3)nc2c1 Homo sapiens CHEMBL3705193 single protein format
CHEMBL3675778 OBDepict H N N N O F F F IC50 = 1000.0 nM 279.22 FC(F)(F)Oc1ccc2nc(-c3ccccn3)[nH]c2c1 Homo sapiens CHEMBL3705193 single protein format
CHEMBL3675787 OBDepict H N N N N O IC50 = 1000.0 nM 280.33 c1ccc(-c2nc3ccc(N4CCOCC4)cc3[nH]2)nc1 Homo sapiens CHEMBL3705193 single protein format
CHEMBL3675795 OBDepict CH 3 O N N N H HO IC50 = 1000.0 nM 255.28 COc1ccnc(-c2nc3ccc(CO)cc3[nH]2)c1 Homo sapiens CHEMBL3705193 single protein format