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Q15561 | TEAD4_HUMAN | Transcriptional enhancer factor TEF-3 (TEAD4)

3D structures mapped by conservation among orthologs

[ Domain: "tri-helical" // TEA ]

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[ Domain: "Immunoglobulin/Fibronectin type III/E set domains/PapD-like" // KOG3841 ]

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[ Alpha Fold Model ] (go)


Known binders annotated in ChEMBL

IC50 table

molecule_chembl_id structure assay_type relation values units mol_wt smiles organism assay_chembl_id bao_label
CHEMBL242708 OBDepict OH O O OH N H IC50 = 70.0 nM 323.35 O=c1cc(CO)oc(C(Nc2ccccc2)c2ccccc2)c1O Homo sapiens CHEMBL4670810 cell-based format
CHEMBL4459587 OBDepict CH 2 S NH O O IC50 = 197.0 nM 323.42 C=CS(=O)(=O)Nc1ccc(Cc2ccc3ccccc3c2)cc1 Homo sapiens CHEMBL4378772 cell-based format