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Q6SZW1 | SARM1_HUMAN | NAD(+) hydrolase SARM1 (SARM1)

3D structures mapped by conservation among orthologs

[ Domain: "SAM domain-like" // SAM_1 ]

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[ Domain: "Toll/Interleukin receptor TIR domain" // TIR ]

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[ Domain: pdbs with more than 2 multi-domains ]

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[ Alpha Fold Model ] (go)


Known binders annotated in ChEMBL

IC50 table

molecule_chembl_id structure assay_type relation values units mol_wt smiles organism assay_chembl_id bao_label
CHEMBL2009370 OBDepict CH 3 N CH 3 S N S N O IC50 = 150.0 nM 241.34 CN(C)c1n/c(=N/Cc2ccco2)ss1 Homo sapiens CHEMBL4422590 cell-based format
CHEMBL2004241 OBDepict H 3 C N H 3 C S N S N O BrH IC50 < 150.0 nM 322.25 Br.CN(C)c1n/c(=N/Cc2ccco2)ss1 Homo sapiens CHEMBL4422580 cell-based format
CHEMBL2009483 OBDepict Cl N S N S N CH 3 H 3 C IC50 = 700.0 nM 271.8 CN(C)c1n/c(=N/c2cccc(Cl)c2)ss1 Homo sapiens CHEMBL4422590 cell-based format