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Q86U86 | PB1_HUMAN | Protein polybromo-1 (PBRM1)

3D structures mapped by conservation among orthologs

[ Domain: "Bromodomain" // Bromodomain ]

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[ Alpha Fold Model ] (go)


Known binders annotated in ChEMBL

IC50 table

molecule_chembl_id structure assay_type relation values units mol_wt smiles organism assay_chembl_id bao_label
CHEMBL4650213 OBDepict O HO N H H N N IC50 = 550.3 nM 321.38 O=C(C=CN1C[C@H]2C[C@@H]1CN2c1ccccn1)c1ccccc1O Homo sapiens CHEMBL4650019 single protein format