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Q8N5Y8 | PAR16_HUMAN | Protein mono-ADP-ribosyltransferase PARP16 (PARP16)

3D structures mapped by conservation among orthologs

[ Domain: "ADP-ribosylation" // PARP ]

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[ Domain: "Domain of poly(ADP-ribose) polymerase" // EUF08131 ]

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[ Domain: pdbs with more than 2 multi-domains ]

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[ Alpha Fold Model ] (go)


Known binders annotated in ChEMBL

IC50 table

molecule_chembl_id structure assay_type relation values units mol_wt smiles organism assay_chembl_id bao_label
CHEMBL4089522 OBDepict O NH N O O NH 2 N F IC50 = 560.0 nM 396.42 NC(=O)c1cccc(NC(=O)/C=CC(=O)N2CCN(c3ccc(F)cc3)CC2)c1 Homo sapiens CHEMBL4022070 single protein format