Q8WTS6 | SETD7_HUMAN | Histone-lysine N-methyltransferase SETD7 (SETD7)
3D structures mapped by conservation among orthologs
[ Domain: "SET domain-like" // SET ]
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[ Domain: "Histone H3 K4-specific methyltransferase SET7/9-N" // KOG1079_3rd_1 ]
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[ Alpha Fold Model ] (go)
Known binders annotated in ChEMBL
IC50 table
| molecule_chembl_id | structure | assay_type | relation | values | units | mol_wt | smiles | organism | assay_chembl_id | bao_label |
|---|---|---|---|---|---|---|---|---|---|---|
| CHEMBL3414622 | IC50 | = | 2.0 | nM | 499.53 | O=C([C@@H](Cc1cccc(C(F)(F)F)c1)NS(=O)(=O)c1cc(F)c2c(c1)CCNC2)N1CCCC1 | Homo sapiens | CHEMBL3420688 | assay format | |
| CHEMBL516 | IC50 | = | 1000.0 | nM | 287.41 | CN1CCC(=C2c3ccccc3C=Cc3ccccc32)CC1 | Homo sapiens | CHEMBL3812774 | assay format |