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Q92830 | KAT2A_HUMAN | Histone acetyltransferase KAT2A (KAT2A)

3D structures mapped by conservation among orthologs

[ Domain: "Acyl-CoA N-acyltransferases (Nat)" // Acetyltransf_10 ]

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[ Domain: "Bromodomain" // Bromodomain ]

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[ Domain: pdbs with more than 2 multi-domains ]

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[ Alpha Fold Model ] (go)


Known binders annotated in ChEMBL

Ki table

molecule_chembl_id structure assay_type relation values units mol_wt smiles organism assay_chembl_id bao_label
CHEMBL4069412 OBDepict CH 3 N H N H H N Br N O CH 3 Ki = 1.4 nM 377.29 CN1C[C@H](Nc2cnn(C)c(=O)c2Br)C[C@H](c2ccccc2)C1 Homo sapiens CHEMBL4003548 assay format