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Q96B36 | AKTS1_HUMAN | Proline-rich AKT1 substrate 1 (AKT1S1)

3D structures mapped by conservation among orthologs



[ Alpha Fold Model ] (go)


Known binders annotated in ChEMBL

IC50 table

molecule_chembl_id structure assay_type relation values units mol_wt smiles organism assay_chembl_id bao_label
CHEMBL1257282 OBDepict F NH 2 H N O N N N H 3 C N H IC50 = 160.0 nM 382.44 Cc1c[nH]c2ncnc(N3CCN(C(=O)[C@H](N)Cc4ccc(F)cc4)CC3)c12 Homo sapiens CHEMBL1259577 cell-based format