HOME LIGAND hPROTEOME OTHERS DOCUMENT

Q9BVS4 | RIOK2_HUMAN | Serine/threonine-protein kinase RIO2 (RIOK2)

3D structures mapped by conservation among orthologs

[ Domain: "winged" // Rio2_N ]

download pymol session

[ Domain: "Protein kinase" // RIO1 ]

download pymol session

[ Domain: pdbs with more than 2 multi-domains ]

download pymol session



[ Alpha Fold Model ] (go)


Known binders annotated in ChEMBL

IC50 table

molecule_chembl_id structure assay_type relation values units mol_wt smiles organism assay_chembl_id bao_label
CHEMBL4858983 OBDepict CH 3 S O O HO HO N N N CH 3 CH 3 N IC50 = 130.0 nM 338.39 CN(C)c1ccc(/N=N/c2ccccn2)c(O)c1.CS(=O)(=O)O Homo sapiens CHEMBL4825563 cell-based format