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Q9UBS5 | GABR1_HUMAN | Gamma-aminobutyric acid type B receptor subunit 1 (GABBR1)

3D structures mapped by conservation among orthologs

[ Domain: "Periplasmic binding protein-like I" // ANF_receptor_2nd ]

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[ Domain: "Periplasmic binding protein-like I" // ANF_receptor_2nd_1 ]

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[ Domain: "Complement control module/SCR domain" // Sushi_3 ]

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[ Alpha Fold Model ] (go)


Known binders annotated in ChEMBL

IC50 table Ki table

molecule_chembl_id structure assay_type relation values units mol_wt smiles organism assay_chembl_id bao_label
CHEMBL2391908 OBDepict Cl Cl N H CH 3 H OH H P O OH ClH Ki = 2.9 nM 444.77 C[C@H](NC[C@H](O)CP(=O)(O)CC1CCCCC1)c1ccc(Cl)c(Cl)c1.Cl Homo sapiens CHEMBL2395266 cell-based format
CHEMBL2391908 OBDepict Cl Cl N H CH 3 H OH H P O OH ClH IC50 = 6.4 nM 444.77 C[C@H](NC[C@H](O)CP(=O)(O)CC1CCCCC1)c1ccc(Cl)c(Cl)c1.Cl Homo sapiens CHEMBL2395266 cell-based format