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Q9Y253 | POLH_HUMAN | DNA polymerase eta (POLH)

3D structures mapped by conservation among orthologs

[ Domain: "SAM domain-like" // KOG2095_1st ]

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[ Domain: "Lesion bypass DNA polymerase (Y-family), little finger domain" // IMS_C ]

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[ Domain: "Adenylyl and guanylyl cyclase catalytic domain-like" // IMS ]

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[ Domain: "beta-beta-alpha zinc fingers" // KOG2095_2nd ]

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[ Domain: "Hypothetical protein Ta1206-like" // IMS_1 ]

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[ Domain: pdbs with more than 2 multi-domains ]

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[ Alpha Fold Model ] (go)


Known binders annotated in ChEMBL

IC50 table

molecule_chembl_id structure assay_type relation values units mol_wt smiles organism assay_chembl_id bao_label
CHEMBL6246 OBDepict HO HO O O O O OH OH IC50 = 62.0 nM 302.19 O=c1oc2c(O)c(O)cc3c(=O)oc4c(O)c(O)cc1c4c23 Homo sapiens CHEMBL3854639 assay format
CHEMBL275938 OBDepict OH O O OH HO O OH O HO IC50 = 75.0 nM 422.35 O=C(O)C1=CC(=C(c2ccc(O)c(C(=O)O)c2)c2ccc(O)c(C(=O)O)c2)C=CC1=O Homo sapiens CHEMBL3854639 assay format