Q9Y263 | PLAP_HUMAN | Phospholipase A-2-activating protein (PLAA)
3D structures mapped by conservation among orthologs
[ Domain: "ARM repeat" // PUL ]
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[ Domain: "ubiquitin-binding domain from PLAA" // PFU ]
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[ Alpha Fold Model ] (go)
Known binders annotated in ChEMBL
IC50 table
| molecule_chembl_id | structure | assay_type | relation | values | units | mol_wt | smiles | organism | assay_chembl_id | bao_label |
|---|---|---|---|---|---|---|---|---|---|---|
| CHEMBL1077979 | IC50 | = | 11.0 | nM | 362.38 | COc1cc(O)c2c(c1)/C=C/C[C@H](O)[C@H](O)C(=O)/C=CC[C@H](C)OC2=O | Homo sapiens | CHEMBL4024851 | single protein format | |
| CHEMBL4068569 | IC50 | = | 36.0 | nM | 380.37 | COc1cc(O)c2c(c1)/C=C/C[C@H](O)[C@H](O)C(=O)/C(F)=CC[C@H](C)OC2=O | Homo sapiens | CHEMBL4024851 | single protein format | |
| CHEMBL608723 | IC50 | = | 800.0 | nM | 268.27 | O=C(Cn1cnc2ccccc21)c1ccc(O)c(O)c1 | Homo sapiens | CHEMBL1074487 | single protein format | |
| CHEMBL607856 | IC50 | = | 800.0 | nM | 246.27 | CCc1nccn1CC(=O)c1ccc(O)c(O)c1 | Homo sapiens | CHEMBL1074487 | single protein format |